Formylmelphalan was approved in China for treating cancer. Formylmelphalan is an alkylating agents, which could cross-link DNA.
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Chemical |
CAS Num |
7789-59-5 |
Chemical Formula |
C14H18Cl2N2O3 |
Molecular Weight |
333.21 |
IUPAC Chemical Name |
3-[4-[bis(2-chloroethyl)amino]phenyl]-2-formamidopropanoic acid |
Exact Mass |
332.06945 |
Elemental Analysis |
C, 50.46; H, 5.44; Cl, 21.28; N, 8.41; O, 14.40 |
Synonym |
NFormylmelphalan; NFormylLsarcolysin; NFormylLpsarcolysin; CB 3208; NSC 37024; NSC37024; LS15879. |
Solubility |
Soluble in DMSO, not in water |
SMILES Code |
O=C(O)C(NC=O)CC1=CC=C(N(CCCl)CCCl)C=C1 |
Biological |
Targets and Effects |
N/A |
Pathways |
alkylating agent |
Physical |
Appearance |
Solid powder |
Purity |
>98% (or refer to the Certificate of Analysis) |
Shipping Condition |
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
Storage Condition |
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
Shelf Life |
>2 years if stored properly |